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PharmacyMedicinal ChemistryPharmacologyDrug DesignMolecular PharmacologyStructure-activity RelationshipsDrug-receptor InteractionsEnzyme InhibitionHeterocyclic ChemistryLead Compound DesignLigand BindingStructure-activity Relationship AnalysisHeterocyclic Medicinal ChemistryMedicinal HeterocyclesPyrazole ChemistryStructure-activity Relationship Modeling
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Thomas D. Penning, John J. Talley, Stephen R. Bertenshaw et al. · Journal of Medicinal Chemistry · 1997 · 2K citations · Full text
Structural basis for selective inhibition of cyclooxygenase-2 by anti-inflammatory agents
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