Andrei Shavnya

Palladium-Catalyzed Sulfination of Aryl and Heteroaryl Halides: Direct Access to Sulfones and Sulfonamides

Andrei Shavnya, Steven B. Coffey, Aaron Smith et al. · Organic Letters · 2013 · 225 citations

Chemical Engineering, Cross-coupling Reaction, Engineering +15

Discovery of PF-04449913, a Potent and Orally Bioavailable Inhibitor of Smoothened

Michael J. Munchhof, Qifang Li, Andrei Shavnya et al. · ACS Medicinal Chemistry Letters · 2011 · 158 citations · Full text

Pharmaceutical Science, Chemoprevention Strategy, Smoothened Inhibitor +20

Synthesis of Sulfones from Organozinc Reagents, DABSO, and Alkyl Halides

Benjamin N. Rocke, Kevin B. Bahnck, Michael Herr et al. · Organic Letters · 2013 · 152 citations

Medicinal Chemistry, So2 Surrogate Dabso, Zinc Sulfinate Salts +11

5-Heteroatom substituted pyrazoles as canine COX-2 inhibitors. Part 1: Structure–activity relationship studies of 5-alkylamino pyrazoles and discovery of a potent, selective, and orally active analog

Subas M. Sakya, Kristin M. Lundy DeMello, Martha L. Minich et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 51 citations · Full text

5-Alkylamino Pyrazoles, Molecular Pharmacology, Medicinal Chemistry +11

Discovery of a potent, selective and orally active canine COX-2 inhibitor, 2-(3-difluoromethyl-5-phenyl-pyrazol-1-yl)-5-methanesulfonyl-pyridine

Jin Li, Kristin M. Lundy DeMello, Henry S. Cheng et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 38 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Medicine +7