Concepedia

Pyridyl-pyrimidine benzimidazole derivatives as potent, selective, and orally bioavailable inhibitors of Tie-2 kinase

Victor J. Cee, Alan C. Cheng, Karina Romero, S.F. Bellon, Christopher Mohr, Douglas A. Whittington, Annette Bak, James Bready, Sean Caenepeel, Angela Coxon,

Bioorganic & Medicinal Chemistry Letters · 2008 · 64 citations · 10 references

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10

Structure of the Tie2 RTK Domain

Lisa M. Shewchuk, Anne M. Hassell, Byron Ellis et al. · Structure · 2000 · 145 citations · Full text

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Ablation of the spindle assembly checkpoint by a compound targeting Mps1

Marc Schmidt, Yemima Budirahardja, Rob Klompmaker et al. · EMBO Reports · 2005 · 115 citations · Full text

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Mitotic requirement for aurora A kinase is bypassed in the absence of aurora B kinase

Hui Yang, Teresa F. Burke, Jack Dempsey et al. · FEBS Letters · 2005 · 114 citations

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Evolution of a Highly Selective and Potent 2-(Pyridin-2-yl)-1,3,5-triazine Tie-2 Kinase Inhibitor

Brian L. Hodous, Stephanie Geuns-Meyer, Paul E. Hughes et al. · Journal of Medicinal Chemistry · 2007 · 91 citations · Full text

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Di-2-Pyridyl thionocarbonate. A new reagent for the preparation of isothiocyanates and carbodiimides.

Sunggak Kim, Kyu Yang Yi · Tetrahedron Letters · 1985 · 81 citations

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