Concepedia

Concept

lead optimization

Parents

383

Publications

31.5K

Citations

3K

Authors

483

Institutions

About

Lead optimization is an iterative process in drug discovery and development focused on systematically improving the pharmacological, pharmacokinetic, and toxicological properties of initial biologically active compounds or 'leads' through structural modification and rigorous evaluation to identify viable drug candidates.

Top Authors

Rankings shown are based on concept H-Index.

EN

University of Naples Federico II

JB

University of Bonn

SJ

GlaxoSmithKline (United Kingdom)

LM

University of Naples Federico II

SC

University of Naples Federico II

Top Institutions

Rankings shown are based on concept H-Index.

AstraZeneca (United Kingdom)

Cambridge, United Kingdom

Pfizer (United States)

New York, United States

Bayer (Germany)

Leverkusen, Germany

GlaxoSmithKline (United Kingdom)

London, United Kingdom