Concepedia

Mining Public Domain Data to Develop Selective DYRK1A Inhibitors

Scott H. Henderson, F.J. Sorrell, James M. Bennett, Marcus T. Hanley, Sean W. Robinson, Iva Navrátilová, Jonathan M. Elkins, Simon E. Ward

ACS Medicinal Chemistry Letters · 2020 · 17 citations · 22 references

DOIFull text

Open access

Concepts

Abstract

, a highly selective DYRK1A inhibitor.

References

22

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KNIME - the Konstanz information miner

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Moving beyond Rules: The Development of a Central Nervous System Multiparameter Optimization (CNS MPO) Approach To Enable Alignment of Druglike Properties

Travis T. Wager, Xinjun Hou, Patrick R. Verhoest et al. · ACS Chemical Neuroscience · 2010 · 1K citations

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