Concepedia

Discovery, Characterization, and Antiparkinsonian Effect of Novel Positive Allosteric Modulators of Metabotropic Glutamate Receptor 4

Colleen M. Niswender, Kari A. Johnson, C. David Weaver, Carrie K. Jones, Zixiu Xiang, Qingwei Luo, Alice L. Rodriguez, Joy E. Marlo, Tomas de Paulis, Analisa D. Thompson,

Molecular Pharmacology · 2008 · 186 citations · 27 references

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References

27

Substitution of three amino acids switches receptor specificity of Gqα to that of Giα

Bruce R. Conklin, Zvi Farfel, Kevin D. Lustig et al. · Nature · 1993 · 736 citations

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Ro 25–6981, a Highly Potent and Selective Blocker of N-Methyl-d-aspartate Receptors Containing the NR2B Subunit. Characterization in Vitro

G. Fischer, Vincent Mutel, Gerhard Trube et al. · Journal of Pharmacology and Experimental Therapeutics · 1997 · 484 citations

, , +17

A Novel Selective Positive Allosteric Modulator of Metabotropic Glutamate Receptor Subtype 5 Has in Vivo Activity and Antipsychotic-Like Effects in Rat Behavioral Models

Gene G. Kinney, Julie A. O’Brien, Wei Lemaire et al. · Journal of Pharmacology and Experimental Therapeutics · 2005 · 299 citations

, , +17

Allosteric modulation of group III metabotropic glutamate receptor 4: A potential approach to Parkinson's disease treatment

Michael J. Marino, David L. Williams, Julie A. O’Brien et al. · Proceedings of the National Academy of Sciences · 2003 · 237 citations · Full text

, , +17

Cloning and Expression of Rat Metabotropic Glutamate Receptor 8 Reveals a Distinct Pharmacological Profile

Julie A. Saugstad, J. Mark Kinzie, Michi M. Shinohara et al. · Molecular Pharmacology · 1997 · 205 citations

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