Concepedia

Design and synthesis of novel pyrimido[4,5-b]azepine derivatives as HER2/EGFR dual inhibitors

Youichi Kawakita, Masaki Seto, Tomohiro Ohashi, Toshiya Tamura, Tadashi Yusa, Hiroshi Miki, Hidehisa Iwata, Hidenori Kamiguchi, Toshimasa Tanaka, Satoshi Sogabe,

Bioorganic & Medicinal Chemistry · 2013 · 76 citations · 31 references

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31

[20] Processing of X-ray diffraction data collected in oscillation mode

Zbyszek Otwinowski, W. Minor · Methods in enzymology on CD-ROM/Methods in enzymology · 1997 · 33.6K citations

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<i>MOLREP</i>: an Automated Program for Molecular Replacement

A. A. Vagin, A. Teplyakov · Journal of Applied Crystallography · 1997 · 4.8K citations

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Crystal structures of the kinase domain of c-Abl in complex with the small molecule inhibitors PD173955 and imatinib (STI-571).

Bhushan Nagar, William G. Bornmann, Patricia Pellicena et al. · PubMed · 2002 · 941 citations

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Structural Analysis of the Mechanism of Inhibition and Allosteric Activation of the Kinase Domain of HER2 Protein

Kathleen Aertgeerts, R.J. Skene, Jason K. Yano et al. · Journal of Biological Chemistry · 2011 · 431 citations · Full text

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The erbB gene of avian erythroblastosis virus is a member of the src gene family

Tadashi Yamamoto, Tsutomu Nishida, Nobuyuki Miyajima et al. · Cell · 1983 · 378 citations

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