Youichi Kawakita

Design and Synthesis of Novel Human Epidermal Growth Factor Receptor 2 (HER2)/Epidermal Growth Factor Receptor (EGFR) Dual Inhibitors Bearing a Pyrrolo[3,2-<i>d</i>]pyrimidine Scaffold

Tomoyasu Ishikawa, Masaki Seto, Hiroshi Banno et al. · Journal of Medicinal Chemistry · 2011 · 207 citations · Full text

Dual Inhibitors Bearing, Medicinal Chemistry, Dual Inhibitors +12

Structure-Based Approach for the Discovery of Pyrrolo[3,2-<i>d</i>]pyrimidine-Based EGFR T790M/L858R Mutant Inhibitors

Satoshi Sogabe, Youichi Kawakita, S. Igaki et al. · ACS Medicinal Chemistry Letters · 2012 · 161 citations · Full text

Molecular Biology, Egfr Inhibitors, Chemical Biology +19

Design and synthesis of novel pyrimido[4,5-b]azepine derivatives as HER2/EGFR dual inhibitors

Youichi Kawakita, Masaki Seto, Tomohiro Ohashi et al. · Bioorganic & Medicinal Chemistry · 2013 · 72 citations · Full text

Design and Synthesis of Pyrrolo[3,2-<i>d</i>]pyrimidine Human Epidermal Growth Factor Receptor 2 (HER2)/Epidermal Growth Factor Receptor (EGFR) Dual Inhibitors: Exploration of Novel Back-Pocket Binders

Youichi Kawakita, Hiroshi Banno, Tomohiro Ohashi et al. · Journal of Medicinal Chemistry · 2012 · 42 citations · Full text

Discovery of Novel and Potent Stearoyl Coenzyme A Desaturase 1 (SCD1) Inhibitors as Anticancer Agents

Keisuke Imamura, Naoki Tomita, Youichi Kawakita et al. · Bioorganic & Medicinal Chemistry · 2017 · 35 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +9