Stanley Kupchinsky

Discovery and SAR of 2-aminothiazole inhibitors of cyclin-dependent kinase 5/p25 as a potential treatment for Alzheimer’s disease

Christopher J. Helal, Mark A. Sanner, Christopher B. Cooper et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 99 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

A novel class of achiral seco-analogs of CC-1065 and the duocarmycins: design, synthesis, DNA binding, and anticancer properties

Stanley Kupchinsky, Sara Centioni, Tiffany T. Howard et al. · Bioorganic & Medicinal Chemistry · 2004 · 21 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

Design, synthesis, and biological evaluation of novel human 5′-deoxy-5′-methylthioadenosine phosphorylase (MTAP) substrates

Pei‐Pei Kung, Luke R. Zehnder, Jerry Meng et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 21 citations

Pharmacy, Biochemistry, Medicinal Chemistry +14

Novel platinum(II) derivatives of analogues of netropsin and distamycin: Synthesis, DNA binding and cytotoxic properties

Moses Lee, Jacob E. Simpson, Adrienne J. Burns et al. · UCL Discovery (University College London) · 1996 · 12 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

N-(Pyridin-2-yl) arylsulfonamide inhibitors of 11β-hydroxysteroid dehydrogenase type 1: Strategies to eliminate reactive metabolites

Sajiv K. Nair, Jean Matthews, Stephan J. Cripps et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 11 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10