Concepedia

A 6-alkylsalicylate histone acetyltransferase inhibitor inhibits histone acetylation and pro-inflammatory gene expression in murine precision-cut lung slices

Thea van den Bosch, Niek G.J. Leus, Hannah Wapenaar, Alexander P. Boichenko, Jos Hermans, Rainer Bischoff, Hidde J. Haisma, Frank J. Dekker

Pulmonary Pharmacology & Therapeutics · 2017 · 25 citations · 22 references

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22

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Substrate and Functional Diversity of Lysine Acetylation Revealed by a Proteomics Survey

Sung Chan Kim, Robert W. Sprung, Yue Chen et al. · Molecular Cell · 2006 · 1.5K citations · Full text

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Molecular Evolution of the Histone Deacetylase Family: Functional Implications of Phylogenetic Analysis

IvanV Gregoretti, Yunmi Lee, Holly V. Goodson · Journal of Molecular Biology · 2004 · 1.5K citations

, , +14

Small Molecule Modulators of Histone Acetyltransferase p300

Karanam Balasubramanyam, Anupama Ranganathan, Tapas K. Kundu · Journal of Biological Chemistry · 2003 · 511 citations · Full text

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A Human Protein Complex Homologous to the <i>Drosophila</i> MSL Complex Is Responsible for the Majority of Histone H4 Acetylation at Lysine 16

Edwin R. Smith, Christelle Cayrou, Rong Huang et al. · Molecular and Cellular Biology · 2005 · 335 citations · Full text

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