Molecular Cell · 2015 · 159 citations · 43 references
Life SciencesGeneticsMolecular BiologyChromatin BiologyChromatin StructureEpigeneticsChromatinChromatin ArchitectureChromatin InteractionsHistone ModificationsHistone ProteinsNucleosome StructureAdaptor Protein RecruitmentChromatin Remodeler Activity
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Selective inhibition of BET bromodomains
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BET Bromodomain Inhibition as a Therapeutic Strategy to Target c-Myc
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RNAi screen identifies Brd4 as a therapeutic target in acute myeloid leukaemia
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Suppression of inflammation by a synthetic histone mimic
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Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia
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