S. Picaud

Selective inhibition of BET bromodomains

P. Filippakopoulos, Jun Qi, S. Picaud et al. · Nature · 2010 · 4.2K citations · Full text

Bet Bromodomains, Genetics, Pathogenesis +3

Histone Recognition and Large-Scale Structural Analysis of the Human Bromodomain Family

P. Filippakopoulos, S. Picaud, Maria Mangos et al. · Cell · 2012 · 1.7K citations · Full text

Structural Bioinformatics, Epigenetic Change, Genetics +25

RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain

S. Picaud, Christopher Wells, I. Felletar et al. · Proceedings of the National Academy of Sciences · 2013 · 475 citations · Full text

Small-Molecule Inhibition of BRDT for Male Contraception

Martin M. Matzuk, Michael R. McKeown, P. Filippakopoulos et al. · Cell · 2012 · 410 citations · Full text

Spermatogenesis, Contraceptive Use, Testis Boundary +24

Dual kinase-bromodomain inhibitors for rationally designed polypharmacology

Pietro Ciceri, Susanne Müller, Alison O’Mahony et al. · Nature Chemical Biology · 2014 · 347 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Medicine +6