Publication | Closed Access
The structure based design of dual HDAC/BET inhibitors as novel epigenetic probes
73
Citations
31
References
2014
Year
Epigenetic ChangeMolecular BiologyEpigeneticsNucleic Acid BiomarkersTumor BiologyNovel Epigenetic ProbesMolecular EpigeneticsProteomicsCell SignalingDual Hdac/bet InhibitorsProtein FunctionBiochemistryCancer CellsTranslational ProteomicsCell BiologyInhibits BetChromatinNatural SciencesEpigenomicsMolecular BasisHdac ProteinsCellular BiochemistryMedicineGenome EditingDrug Discovery
DUAL946 (1) inhibits BET and HDAC proteins in chemoproteomic cell lysate experiments and in immune and cancer cells.
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