Concepedia

Imidazo[1,2-a]pyridin-3-amines as potential HIV-1 non-nucleoside reverse transcriptase inhibitors

Moira L. Bode, David Gravestock, Simon S. Moleele, Christiaan W. van der Westhuyzen, Stephen C. Pelly, Paul A. Steenkamp, Heinrich C. Hoppe, Tasmiyah Khan, Lindiwe A. Nkabinde

Bioorganic & Medicinal Chemistry · 2011 · 114 citations · 17 references

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17

Atomic Physicochemical Parameters for Three‐Dimensional Structure‐Directed Quantitative Structure‐Activity Relationships I. Partition Coefficients as a Measure of Hydrophobicity

Arup K. Ghose, Gordon M. Crippen · Journal of Computational Chemistry · 1986 · 627 citations · Full text

, , +17

Synthesis of Imidazo[1,2-a] annulated Pyridines, Pyrazines and Pyrimidines by a Novel Three-Component Condensation

Katrin Groebke, Lutz Weber, Fridolin Mehlin · Synlett · 1998 · 430 citations

, , +9

Parallel synthesis of 3-aminoimidazo[1,2-a]pyridines and pyrazines by a new three-component condensation

Christopher Blackburn, Bing Guan, Paul Fleming et al. · Tetrahedron Letters · 1998 · 371 citations

, , +12

Crystal Structures of HIV-1 Reverse Transcriptase with Etravirine (TMC125) and Rilpivirine (TMC278): Implications for Drug Design

E.B. Lansdon, Katherine M. Brendza, Magdeleine Hung et al. · Journal of Medicinal Chemistry · 2010 · 226 citations

, , +17

Synthesis of Imidazo[1,2-<i>a</i>]pyridines as Antiviral Agents

Alain Gueiffier, Sylvie Mavel, Mohammed Lhassani et al. · Journal of Medicinal Chemistry · 1998 · 217 citations

, , +16