Concepedia

Activity probe for in vivo profiling of the specificity of proteasome inhibitor bortezomib

Celia R. Berkers, Martijn Verdoes, Eben I. Lichtman, Edda Fiebiger, Benedikt M. Kessler, Kenneth C. Anderson, Hidde L. Ploegh, Huib Ovaa, Paul J. Galardy

Nature Methods · 2005 · 266 citations · 19 references

DOI

Concepts

References

19

The proteasome inhibitor PS-341 inhibits growth, induces apoptosis, and overcomes drug resistance in human multiple myeloma cells.

Teru Hideshima, Paul G. Richardson, D Chauhan et al. · PubMed · 2001 · 1.5K citations

, , +17

Proteasome inhibitors: a novel class of potent and effective antitumor agents.

Julian Adams, Vito J. Palombella, Edward A. Sausville et al. · PubMed · 1999 · 1.5K citations

, , +14

Activity-based protein profiling: The serine hydrolases

Yongsheng Liu, Matthew P. Patricelli, Benjamin F. Cravatt · Proceedings of the National Academy of Sciences · 1999 · 1.1K citations

, , +16

Short-lived green fluorescent proteins for quantifying ubiquitin/proteasome-dependent proteolysis in living cells

Nico P. Dantuma, Kristina Lindsten, Rickard Glas et al. · Nature Biotechnology · 2000 · 617 citations

, , +13

Epoxide electrophiles as activity-dependent cysteine protease profiling and discovery tools

Doron C. Greenbaum, Katalin F. Medzihradszky, Alma L. Burlingame et al. · Chemistry & Biology · 2000 · 584 citations · Full text

, , +16