A platform for designing HIV integrase inhibitors. Part 2: A two-metal binding model as a potential mechanism of HIV integrase inhibitors

The protein data bank: A computer-based archival file for macromolecular structures

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Inhibitors of Strand Transfer That Prevent Integration and Inhibit HIV-1 Replication in Cells

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Diketo acid inhibitor mechanism and HIV-1 integrase: Implications for metal binding in the active site of phosphotransferase enzymes

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Three new structures of the core domain of HIV-1 integrase: An active site that binds magnesium

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A naphthyridine carboxamide provides evidence for discordant resistance between mechanistically identical inhibitors of HIV-1 integrase

Daria J. Hazuda, Neville J. Anthony, Robert Gomez et al. · Proceedings of the National Academy of Sciences · 2004 · 333 citations · Full text

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