Concepedia

Novel (4-Piperidin-1-yl)-phenyl Sulfonamides as Potent and Selective Human β3 Agonists

Baihua Hu, John W. Ellingboe, Stella Han, Elwood Largis, Kitae Lim, Michael S. Malamas, Ruth Mulvey, Chuansheng Niu, Alexander Oliphant, Jeffrey C. Pelletier,

Bioorganic & Medicinal Chemistry · 2001 · 45 citations · 30 references

DOI

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References

30

cDNA for the human beta 2-adrenergic receptor: a protein with multiple membrane-spanning domains and encoded by a gene whose chromosomal location is shared with that of the receptor for platelet-derived growth factor.

Brian K. Kobilka, Richard A. F. Dixon, Thomas Frielle et al. · Proceedings of the National Academy of Sciences · 1987 · 683 citations · Full text

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Time of Onset of Non-Insulin-Dependent Diabetes Mellitus and Genetic Variation in the β<sub>3</sub>-Adrenergic–Receptor Gene

Jeremy Walston, Kristi D. Silver, Clifton Bogardus et al. · New England Journal of Medicine · 1995 · 596 citations · Full text

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Cloning of the cDNA for the human beta 1-adrenergic receptor.

Thomas Frielle, Sheila Collins, Kiefer W. Daniel et al. · Proceedings of the National Academy of Sciences · 1987 · 580 citations · Full text

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Disodium (R,R)-5-[2-[[2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]-1,3-benzodioxole-2,2-dicarboxylate (CL 316,243). A potent .beta.-adrenergic agonist virtually specific for .beta.3 receptors. A promising antidiabetic and antiobesity agent

Jonathan D. Bloom, Minu Dutia, Bernard D. Johnson et al. · Journal of Medicinal Chemistry · 1992 · 297 citations · Full text

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Prospects for beta 3-adrenoceptor agonists in the treatment of obesity and diabetes.

J R Arch, S. Wilson · PubMed · 1996 · 136 citations

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