Michael S. Malamas

Evaluation of fluorescence-based thermal shift assays for hit identification in drug discovery

Mei-Chu Lo, Ann Aulabaugh, Guixian Jin et al. · Analytical Biochemistry · 2004 · 685 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14

Evaluation of an Estrogen Receptor-β Agonist in Animal Models of Human Disease

Heather A. Harris, Leo Albert, Yelena Leathurby et al. · Endocrinology · 2003 · 313 citations · Full text

Medicine, Endocrinology, Pharmacology +17

Quinazolineacetic acids and related analogs as aldose reductase inhibitors

Michael S. Malamas, Jane Millen · Journal of Medicinal Chemistry · 1991 · 278 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8

Phosphodiesterase 10A Inhibitor Activity in Preclinical Models of the Positive, Cognitive, and Negative Symptoms of Schizophrenia

Steven M. Grauer, Virginia Pulito, Rachel L. Navarra et al. · Journal of Pharmacology and Experimental Therapeutics · 2009 · 266 citations

Medicine, Neuroscience, Pharmacology +13

Design and Synthesis of Aryl Diphenolic Azoles as Potent and Selective Estrogen Receptor-β Ligands

Michael S. Malamas, Eric S. Manas, Robert McDevitt et al. · Journal of Medicinal Chemistry · 2004 · 260 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17