Stereoselective synthesis of 2(S)-(1,1-dimethylethylsulfonylmethyl)-3-(1-naphthyl)-propionic acid, building block for protease inhibitors via asymmetric hydrogenation

New Peptide Synthesis

Hans Wissmann, Hanß‐Jerg Kleiner · Angewandte Chemie International Edition in English · 1980 · 182 citations

Natural Sciences, Biochemistry, Synthetic Medicinal Chemistry +2

Synthesis and biological activity of some transition-state inhibitors of human renin

Walter Fuhrer, Vittorio Rasetti, H. Rüeger et al. · Journal of Medicinal Chemistry · 1988 · 111 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Asymmetric hydrogenation of cycloalkanones catalyzed by BINAP-iridium(I)-aminophosphine systems

Xiaoyong Zhang, T. TAKETOMI, Takashi Yoshizumi et al. · Journal of the American Chemical Society · 1993 · 110 citations

Natural Sciences, Biochemistry, Chemistry +10

Chiral poisoning: a novel strategy for asymmetric catalysis

J.W. Faller, J. Parr · Journal of the American Chemical Society · 1993 · 95 citations

Natural Sciences, Chemistry, Biocatalysis +6

Vanadium(<scp>II</scp>)‐ and Niobium(<scp>III</scp>)‐Induced, Diastereoselective Pinacol Coupling of Peptide Aldehydes to <i>C</i>₂‐Symmetrical HIV‐Protease Inhibitors

Bernhard Kammermeier, Gerhard Beck, Heiner Jendralla et al. · Angewandte Chemie International Edition in English · 1994 · 74 citations

Natural Sciences, Chemistry, Medicinal Chemistry +14