Sean R. Bollinger

An insecticide resistance-breaking mosquitocide targeting inward rectifier potassium channels in vectors of Zika virus and malaria

Daniel R. Swale, Darren W. Engers, Sean R. Bollinger et al. · Scientific Reports · 2016 · 80 citations · Full text

Life Sciences, Entomology, Medicinal Chemistry +17

Identification of Positive Allosteric Modulators VU0155094 (ML397) and VU0422288 (ML396) Reveals New Insights into the Biology of Metabotropic Glutamate Receptor 7

Nidhi Jalan‐Sakrikar, Julie R. Field, Rebecca Klar et al. · ACS Chemical Neuroscience · 2014 · 67 citations · Full text

Life Sciences, Neuroscience, Pharmacology +17

Design and Synthesis of <i>N</i>-Aryl Phenoxyethoxy Pyridinones as Highly Selective and CNS Penetrant mGlu₃ NAMs

Julie L. Engers, Katrina A. Bollinger, Rebecca L. Weiner et al. · ACS Medicinal Chemistry Letters · 2017 · 44 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery, Structure–Activity Relationship, and Biological Characterization of a Novel Series of 6-((1<i>H</i>-Pyrazolo[4,3-<i>b</i>]pyridin-3-yl)amino)-benzo[<i>d</i>]isothiazole-3-carboxamides as Positive Allosteric Modulators of the Metabotropic Glutamate Receptor 4 (mGlu₄)

Sean R. Bollinger, Darren W. Engers, Joseph D. Panarese et al. · Journal of Medicinal Chemistry · 2018 · 26 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Discovery and characterization of N-(1,3-dialkyl-1H-indazol-6-yl)-1H-pyrazolo[4,3-b]pyridin-3-amine scaffold as mGlu4 positive allosteric modulators that mitigate CYP1A2 induction liability

Darren W. Engers, Sean R. Bollinger, Julie L. Engers et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 14 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14