Genta Tadano

Discovery of Imidazo[1,2-<i>b</i>]pyridazine Derivatives: Selective and Orally Available Mps1 (TTK) Kinase Inhibitors Exhibiting Remarkable Antiproliferative Activity

Ken‐ichi Kusakabe, Nobuyuki Ide, Yataro Daigo et al. · Journal of Medicinal Chemistry · 2015 · 64 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +13

Pd‐Catalyzed Stereospecific Azide Substitution of α,β‐Unsaturated γ,δ‐Epoxy Esters with Double Inversion of Configuration

Masaaki Miyashita, Taiku Mizutani, Genta Tadano et al. · Angewandte Chemie International Edition · 2005 · 53 citations

Engineering, Amino Acids, δ‐Epoxy Esters +16

Pd‐Catalyzed Stereospecific Azide Substitution of α,β‐Unsaturated γ,δ‐Epoxy Esters with Double Inversion of Configuration

Masaaki Miyashita, Taiku Mizutani, Genta Tadano et al. · Angewandte Chemie · 2005 · 35 citations

Structure-Based Design of Selective β-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors: Targeting the Flap to Gain Selectivity over BACE2

Kazuki Fujimoto, Eriko Matsuoka, Naoya Asada et al. · Journal of Medicinal Chemistry · 2019 · 35 citations · Full text

Drug Target, Protein Assembly, Molecular Biology +17

Diaminopyridine-Based Potent and Selective Mps1 Kinase Inhibitors Binding to an Unusual Flipped-Peptide Conformation

Ken‐ichi Kusakabe, Nobuyuki Ide, Yataro Daigo et al. · ACS Medicinal Chemistry Letters · 2012 · 33 citations · Full text

Molecular Biology, Chemical Biology, Unusual Flipped-peptide Conformation +17