Concepedia

Edward S. Tasber

ES

Statistics

Publications

9

Citations

384

H-Index

9

Active since

2003

Affiliations

United States Military Academy(Current)

Edward S. Tasber is an author at United States Military Academy specializing in drug discovery, enzyme inhibition, and pharmacy.

Publications per year

2003–2008

9

Publications

9

Development of thioquinazolinones, allosteric Chk1 kinase inhibitors

Antonella Converso, Timothy J. Hartingh, R. M. Garbaccio et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 74 citations · Full text

, , +10

Kinesin spindle protein (KSP) inhibitors. Part 2: The design, synthesis, and characterization of 2,4-diaryl-2,5-dihydropyrrole inhibitors of the mitotic kinesin KSP

Mark E. Fraley, R. M. Garbaccio, Kenneth L. Arrington et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 64 citations · Full text

, , +16

Discovery and biochemical characterization of selective ATP competitive inhibitors of the human mitotic kinesin KSP

Keith Rickert, Michael D. Schaber, Maricel Torrent et al. · Archives of Biochemistry and Biophysics · 2007 · 50 citations

, , +16

Kinesin spindle protein (KSP) inhibitors. Part 3: Synthesis and evaluation of phenolic 2,4-diaryl-2,5-dihydropyrroles with reduced hERG binding and employment of a phosphate prodrug strategy for aqueous solubility

R. M. Garbaccio, Mark E. Fraley, Edward S. Tasber et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 47 citations · Full text

, , +17

Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors

Edward J. Brnardic, R. M. Garbaccio, Mark E. Fraley et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 44 citations · Full text

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