Concepedia

Designing an eEF2K-Targeting PROTAC small molecule that induces apoptosis in MDA-MB-231 cells

Yao Liu, Yongqi Zhen, Guan Wang, Gaoxia Yang, Leilei Fu, Bo Liu, Liang Ouyang

European Journal of Medicinal Chemistry · 2020 · 32 citations · 29 references

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29

SWISS-MODEL: homology modelling of protein structures and complexes

Andrew Waterhouse, Martino Bertoni, Stefan Bienert et al. · Nucleic Acids Research · 2018 · 13.6K citations · Full text

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The eEF2 Kinase Confers Resistance to Nutrient Deprivation by Blocking Translation Elongation

Gabriel Leprivier, Marc Remke, Barak Rotblat et al. · Cell · 2013 · 416 citations · Full text

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Light-Induced Protein Degradation with Photocaged PROTACs

Gang Xue, Kun Wang, Danli Zhou et al. · Journal of the American Chemical Society · 2019 · 344 citations

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Structure of the CaMKIIδ/Calmodulin Complex Reveals the Molecular Mechanism of CaMKII Kinase Activation

P. Rellos, A.C.W. Pike, F. Niesen et al. · PLoS Biology · 2010 · 306 citations · Full text

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Addressing Kinase-Independent Functions of Fak via PROTAC-Mediated Degradation

Philipp M. Cromm, Kusal T. G. Samarasinghe, John Hines et al. · Journal of the American Chemical Society · 2018 · 285 citations

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