Concepedia

Conformationally restricted homotryptamines. Part 4: Heterocyclic and naphthyl analogs of a potent selective serotonin reuptake inhibitor

Dalton King, Derek J. Denhart, Jeffrey A. Deskus, Jonathan L. Ditta, James R. Epperson, Mendi A. Higgins, Joyce E. Kung, Lawrence R. Marcin, C.P. Sloan, Gail K. Mattson,

Bioorganic & Medicinal Chemistry Letters · 2007 · 22 citations · 8 references

DOIFull text

Open access

Concepts

References

8

Thiol Ester−Boronic Acid Coupling. A Mechanistically Unprecedented and General Ketone Synthesis

Lanny S. Liebeskind, Jiří Šrogl · Journal of the American Chemical Society · 2000 · 630 citations

, , +6

Enantioselective Synthesis of a Highly Potent Selective Serotonin Reuptake Inhibitor. An Application of Imidazolidinone Catalysis to the Alkylation of Indoles with an α,β-Disubstituted α,β-Unsaturated Aldehyde

Dalton King, Zhaoxing Meng, Derek J. Denhart et al. · Organic Letters · 2005 · 123 citations

, , +17

Synthesis and Structure−Activity Relationship in a Class of Indolebutylpiperazines as Dual 5-HT<sub>1A</sub> Receptor Agonists and Serotonin Reuptake Inhibitors

Timo Heinrich, Henning Böttcher, R. Gericke et al. · Journal of Medicinal Chemistry · 2004 · 116 citations · Full text

, , +17

Conformationally Restricted Homotryptamines. 2. Indole Cyclopropylmethylamines as Selective Serotonin Reuptake Inhibitors

Ronald J. Mattson, John D. Catt, Derek J. Denhart et al. · Journal of Medicinal Chemistry · 2005 · 34 citations · Full text

, , +17

Homotryptamines as potent and selective serotonin reuptake inhibitors (SSRIs)

William D. Schmitz, Derek J. Denhart, Allison B. Brenner et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 26 citations · Full text

, , +10