Concepedia

Discovery of low nanomolar non-hydroxamate inhibitors of tumor necrosis factor-α converting enzyme (TACE)

James J.‐W. Duan, Lihua Chen, Zhonghui Lu, Bin Jiang, Naoyuki Asakawa, James E. Sheppeck, Rui‐Qin Liu, Maryanne Covington, William J. Pitts, Soong‐Hoon Kim,

Bioorganic & Medicinal Chemistry Letters · 2006 · 53 citations · 18 references

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18

Intracellular maturation and localization of the tumour necrosis factor α convertase (TACE)

Johannes Schlöndorff, J. David Becherer, Carl Blobel · Biochemical Journal · 2000 · 353 citations · Full text

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Pyrimidine-2,4,6-Triones: A New Effective and Selective Class of Matrix Metalloproteinase Inhibitors

Frank Grams, Hans Brandstetter, S. D’Alò et al. · Biological Chemistry · 2001 · 142 citations

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The 1.8-Å Crystal Structure of a Matrix Metalloproteinase 8-Barbiturate Inhibitor Complex Reveals a Previously Unobserved Mechanism for Collagenase Substrate Recognition

Hans Brandstetter, Frank Grams, Dagmar Glitz et al. · Journal of Biological Chemistry · 2001 · 127 citations · Full text

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Discovery of γ-Lactam Hydroxamic Acids as Selective Inhibitors of Tumor Necrosis Factor α Converting Enzyme:  Design, Synthesis, and Structure−Activity Relationships

James J.‐W. Duan, Lihua Chen, Zelda R. Wasserman et al. · Journal of Medicinal Chemistry · 2002 · 119 citations · Full text

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Improved method for the Wacker oxidation of cyclic and internal olefins

D. G. Miller, Danial D. M. Wayner · The Journal of Organic Chemistry · 1990 · 116 citations

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