Concepedia

Thiazolidine derivatives as potent and selective inhibitors of the PIM kinase family

Carole J. R. Bataille, Méabh B. Brennan, Simon Byrne, Stephen G. Davies, Matthew J. Durbin, O. Fedorov, K. Huber, Alan M. Jones, Stefan Knapp, Gu Liu,

Bioorganic & Medicinal Chemistry · 2017 · 46 citations · 50 references

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References

50

The use of differential scanning fluorimetry to detect ligand interactions that promote protein stability

F. Niesen, H. Berglund, Masoud Vedadi · Nature Protocols · 2007 · 2.4K citations

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Chemistry: Chemical con artists foil drug discovery

Jonathan B. Baell, Michael A. Walters · Nature · 2014 · 1.1K citations · Full text

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Comprehensive assay of kinase catalytic activity reveals features of kinase inhibitor selectivity

Theonie Anastassiadis, Sean Deacon, Karthik Devarajan et al. · Nature Biotechnology · 2011 · 926 citations · Full text

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Murine leukemia virus-induced T-cell lymphomagenesis: Integration of proviruses in a distinct chromosomal region

H. T. M. Cuypers, Gerard C.M. Selten, Wim Quint et al. · Cell · 1984 · 645 citations

, , +13

In Situ Kinase Profiling Reveals Functionally Relevant Properties of Native Kinases

Matthew P. Patricelli, Tyzoon Nomanbhoy, Jiangyue Wu et al. · Chemistry & Biology · 2011 · 357 citations

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