O. Fedorov

Selective inhibition of BET bromodomains

P. Filippakopoulos, Jun Qi, S. Picaud et al. · Nature · 2010 · 4.2K citations · Full text

Bet Bromodomains, Genetics, Pathogenesis +3

Chemical screening methods to identify ligands that promote protein stability, protein crystallization, and structure determination

Masoud Vedadi, F. Niesen, Abdellah Allali‐Hassani et al. · Proceedings of the National Academy of Sciences · 2006 · 589 citations · Full text

New Ligands, Protein Assembly, Molecular Biology +21

RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain

S. Picaud, Christopher Wells, I. Felletar et al. · Proceedings of the National Academy of Sciences · 2013 · 475 citations · Full text

A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases

O. Fedorov, Brian D. Marsden, Vanda Pogačić et al. · Proceedings of the National Academy of Sciences · 2007 · 375 citations · Full text

Dual kinase-bromodomain inhibitors for rationally designed polypharmacology

Pietro Ciceri, Susanne Müller, Alison O’Mahony et al. · Nature Chemical Biology · 2014 · 347 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Medicine +6