Concepedia

Design and synthesis of selective CDK8/19 dual inhibitors: Discovery of 4,5-dihydrothieno[3′,4′:3,4]benzo[1,2-d]isothiazole derivatives

Koji Ono, Hiroshi Banno, Masanori Okaniwa, Takaharu Hirayama, Naoki Iwamura, Yukiko Hikichi, Saomi Murai, Maki Hasegawa, Yuka Hasegawa, Kazuko Yonemori,

Bioorganic & Medicinal Chemistry · 2017 · 37 citations · 53 references

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References

53

A small molecule–kinase interaction map for clinical kinase inhibitors

Miles A. Fabian, William Biggs, Daniel K. Treiber et al. · Nature Biotechnology · 2005 · 1.9K citations · Full text

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Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

John F. Hartwig · Accounts of Chemical Research · 2008 · 1.9K citations · Full text

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Recent Applications of Palladium‐Catalyzed Coupling Reactions in the Pharmaceutical, Agrochemical, and Fine Chemical Industries

C. Torborg, Matthias Beller · Advanced Synthesis & Catalysis · 2009 · 1.5K citations

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Palladium‐Catalyzed Carbonylation Reactions of Aryl Halides and Related Compounds

Anne Brennführer, Helfried Neumann, Matthias Beller · Angewandte Chemie International Edition · 2009 · 1.4K citations

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Activating RNAs associate with Mediator to enhance chromatin architecture and transcription

Fan Lai, Matteo Cesaroni, Malte Beringer et al. · Nature · 2013 · 860 citations · Full text

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