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Aminoimidazo[1,2-a]pyridines as a new structural class of cyclin-dependent kinase inhibitors. Part 1: Design, synthesis, and biological evaluation

Carlos Jaramillo, J. Eugenio de Diego, Chafiq Hamdouchi, Elizabeth Collins, Heather Keyser, Concha Sánchez-Martı́nez, Miriam Del Prado, Bryan H. Norman, Harold B. Brooks, Scott A. Watkins,

Bioorganic & Medicinal Chemistry Letters · 2004 · 38 citations · 21 references

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Cell cycle control in mammalian cells: role of cyclins, cyclin dependent kinases (CDKs), growth suppressor genes and cyclin-dependent kinase inhibitors (CKIs).

Xavier Graña, E. Premkumar Reddy · PubMed · 1995 · 1.1K citations

Indirubin, the active constituent of a Chinese antileukaemia medicine, inhibits cyclin-dependent kinases

Ralph Hoessel, Sophie Leclerc, Jane Endicott et al. · Nature Cell Biology · 1999 · 811 citations

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Exploiting Chemical Libraries, Structure, and Genomics in the Search for Kinase Inhibitors

Nathanael S. Gray, Lisa Wodicka, A.M.W.H. Thunnissen et al. · Science · 1998 · 806 citations · Full text

Inhibition of Cyclin‐Dependent Kinases by Purine Analogues

Jaroslav Veselý, Libor Havlı́ček, Miroslav Strnad et al. · European Journal of Biochemistry · 1994 · 625 citations · Full text

Inhibition of cyclin-dependent kinases, GSK-3β and CK1 by hymenialdisine, a marine spongeconstituent

Laurent Meijer, A.M.W.H. Thunnissen, AW White et al. · Chemistry & Biology · 2000 · 446 citations · Full text