Scott A. Watkins

Kinetic Characterization of Novel Pyrazole TGF-β Receptor I Kinase Inhibitors and Their Blockade of the Epithelial−Mesenchymal Transition

Sheng-Bin Peng, Lei Yan, Xiaoling Xia et al. · Biochemistry · 2005 · 99 citations

Life Sciences, Cell Biology, Pharmacology +14

Synthesis, Structure−Activity Relationship, and Biological Studies of Indolocarbazoles as Potent Cyclin D1-CDK4 Inhibitors

Guoxin Zhu, Scott E. Conner, Xun Zhou et al. · Journal of Medicinal Chemistry · 2003 · 94 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Structure-based design of a new class of highly selective aminoimidazo[1,2-a]pyridine-based inhibitors of cyclin dependent kinases

Chafiq Hamdouchi, Boyu Zhong, J. S. MENDOZA et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 91 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Novel, potent and selective cyclin D1/CDK4 inhibitors: indolo[6,7-a]pyrrolo[3,4-c]carbazoles

Thomas A. Engler, Kelly Furness, Sushant Malhotra et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 59 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

Aryl[a]pyrrolo[3,4-c]carbazoles as selective cyclin D1-CDK4 inhibitors

Concha Sánchez-Martı́nez, Chuan Shih, Margaret M. Faul et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 53 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10