Bioorganic & Medicinal Chemistry Letters · 2005 · 91 citations · 16 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryStructure-activity RelationshipsChemical Space ExplorationLigand-based DesignMolecular DockingPotency OptimizationStructure-activity Relationship AnalysisCyclin-dependent Kinase 7Cyclin-dependent Kinase 9Kinase Inhibitor Library DesignStructure-activity Relationship Guided DesignStructure-based Lead DiscoveryStructure-based Ligand DesignStructure-based Selectivity Design
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Inhibition of Cyclin‐Dependent Kinases by Purine Analogues
Jaroslav Veselý, Libor Havlı́ček, Miroslav Strnad et al. · European Journal of Biochemistry · 1994 · 626 citations · Full text