J. Eugenio de Diego

The Evolution of High-Throughput Experimentation in Pharmaceutical Development and Perspectives on the Future

Steven M. Mennen, Carolina Alhambra, C. Liana Allen et al. · Organic Process Research & Development · 2019 · 535 citations

Pharmaceutical Research, Pharmaceutical Innovation, Hit Identification +25

Structure-based design of a new class of highly selective aminoimidazo[1,2-a]pyridine-based inhibitors of cyclin dependent kinases

Chafiq Hamdouchi, Boyu Zhong, J. S. MENDOZA et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 90 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Drug Target +12

Aminoimidazo[1,2-a]pyridines as a new structural class of cyclin-dependent kinase inhibitors. Part 1: Design, synthesis, and biological evaluation

Carlos Jaramillo, J. Eugenio de Diego, Chafiq Hamdouchi et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 38 citations · Full text

Combinatorial Chemistry, Cyclin-dependent Kinase Inhibitors, Medicinal Chemistry +11

Regioselective synthesis of 3,6-disubstituted-2-aminoimidazo[1,2-a]pyridines

Carlos Jaramillo, Juan C. Carretero, J. Eugenio de Diego et al. · Tetrahedron Letters · 2002 · 32 citations

Organic Chemistry, Regioselective Synthesis, Synthetic Chemistry +1

The discovery of a new structural class of cyclin-dependent kinase inhibitors, aminoimidazo[1,2-<i>a</i>]pyridines

Chafiq Hamdouchi, Heather Keyser, Elizabeth Collins et al. · Molecular Cancer Therapeutics · 2004 · 29 citations · Full text

Drug Target, Bioorganic Chemistry, Kinase Inhibitors +16