α-Methylation at benzylic fragment of N-aryl-N′-benzyl ureas provides TRPV1 antagonists with better pharmacokinetic properties and higher efficacy in inflammatory pain model

Arthur Gomtsyan, Erol K. Bayburt, Ryan G. Keddy, Sean Turner, Tammie K. Jinkerson, Stanley DiDomenico, Richard J. Perner, John R. Koenig, Irene Drizin, Heath A. McDonald,

Bioorganic & Medicinal Chemistry Letters · 2007 · 33 citations · 10 references

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