Bioorganic & Medicinal Chemistry Letters · 2004 · 33 citations · 5 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryMetabolic StabilityMetabolic Stability EnhancementMetabolic Stability OptimizationPeptidomimetic DesignMetabolic Stability ModulationMetabolic Stability TestingPeptidomimetic Modulators
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Katherine E. Cole, Christine A. Strick, Timothy Paradis et al. · The Journal of Experimental Medicine · 1998 · 879 citations · Full text
The prediction of human clearance from hepatic microsomal metabolism data.