Discovery of a novel class of non-ATP site DFG-out state p38 inhibitors utilizing computationally assisted virtual fragment-based drug design (vFBDD)

Kristofer K. Moffett, Zenon Konteatis, Duyan Nguyen, Rupa Shetty, Jennifer L. Ludington, Ted Fujimoto, Kyoung‐Jin Lee, Xiaomei Chai, H.V.M. Namboodiri, Michael Karpusas,

Bioorganic & Medicinal Chemistry Letters · 2011 · 27 citations · 15 references

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