Bioorganic & Medicinal Chemistry · 2003 · 27 citations · 11 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryStructure-activity RelationshipsCovalent Drug DesignCovalent Inhibitor DesignEnzyme InhibitionLigand BindingLigand-based DesignPotency OptimizationCathepsin ActivityDisulfide Bond ChemistryEnzyme Inhibitor DiscoveryHydrazone LinkersMechanism-based Drug Design
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Vinyl Sulfones as Mechanism-Based Cysteine Protease Inhibitors
James T. Palmer, David Rasnick, Jeffrey L. Klaus et al. · Journal of Medicinal Chemistry · 1995 · 506 citations · Full text
Dieter Brömme, Jeffrey L. Klaus, Kathleen Okamoto et al. · Biochemical Journal · 1996 · 139 citations · Full text