Concepedia

Conformationally constrained farnesoid X receptor (FXR) agonists: Heteroaryl replacements of the naphthalene

Jonathan Y. Bass, Justin A. Caravella, Lihong Chen, Katrina L. Creech, David N. Deaton, Kevin P. Madauss, Harry B. Marr, Robert B. McFadyen, Aaron B. Miller, Wendy Y. Mills,

Bioorganic & Medicinal Chemistry Letters · 2010 · 60 citations · 37 references

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37

Fibroblast growth factor 15 functions as an enterohepatic signal to regulate bile acid homeostasis

Takeshi Inagaki, Mihwa Choi, Antonio Moschetta et al. · Cell Metabolism · 2005 · 1.8K citations · Full text

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A G Protein-coupled Receptor Responsive to Bile Acids

Yuji Kawamata, Ryo Fujii, Masaki Hosoya et al. · Journal of Biological Chemistry · 2003 · 1.6K citations · Full text

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Bile acids lower triglyceride levels via a pathway involving FXR, SHP, and SREBP-1c

Mitsuhiro Watanabe, Sander M. Houten, Li Wang et al. · Journal of Clinical Investigation · 2004 · 1.4K citations · Full text

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Identification of a nuclear receptor that is activated by farnesol metabolites

Barry M. Forman, Elizabeth C. Goode, Jasmine Chen et al. · Cell · 1995 · 1.2K citations · Full text

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Regulation of antibacterial defense in the small intestine by the nuclear bile acid receptor

Takeshi Inagaki, Antonio Moschetta, Youn-Kyoung Lee et al. · Proceedings of the National Academy of Sciences · 2006 · 1.2K citations · Full text

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