Concepedia

Aminopyrrolidineamide inhibitors of site-1 protease

Bruce A. Hay, Barbara Abrams, A Zumbrunn, James J. Valentine, Laurie C. Warren, Stephen F. Petras, Lorraine D. Shelly, Angela Xia, Alison H. Varghese, Julie L. Hawkins,

Bioorganic & Medicinal Chemistry Letters · 2007 · 87 citations · 7 references

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7

Isozyme-nonselective N-Substituted Bipiperidylcarboxamide Acetyl-CoA Carboxylase Inhibitors Reduce Tissue Malonyl-CoA Concentrations, Inhibit Fatty Acid Synthesis, and Increase Fatty Acid Oxidation in Cultured Cells and in Experimental Animals

H. James Harwood, Stephen F. Petras, Lorraine D. Shelly et al. · Journal of Biological Chemistry · 2003 · 243 citations · Full text

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Decreased lipid synthesis in livers of mice with disrupted Site-1 protease gene

Jian Yang, Joseph L. Goldstein, Robert E. Hammer et al. · Proceedings of the National Academy of Sciences · 2001 · 241 citations · Full text

, , +16

Cholic acid mediates negative feedback regulation of bile acid synthesis in mice

Jia Li-Hawkins, Mats Gåfvels, Maria Olin et al. · Journal of Clinical Investigation · 2002 · 227 citations

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Cholic acid mediates negative feedback regulation of bile acid synthesis in mice

Jia Li-Hawkins, Mats Gåfvels, Maria Olin et al. · Journal of Clinical Investigation · 2002 · 225 citations · Full text

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Kinetics of low-density lipoprotein receptor activity in Hep-G2 cells: derivation and validation of a Briggs–Haldane-based kinetic model for evaluating receptor-mediated endocytotic processes in which receptors recycle

H. James Harwood, Lorraine D. Pellarin · Biochemical Journal · 1997 · 35 citations · Full text

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