Concepedia

Design of a series of bicyclic HIV-1 integrase inhibitors. Part 1: Selection of the scaffold

E. D. Jones, Nick Vandegraaff, Giang Le, Neil Choi, William Issa, Katherine Macfarlane, Neeranat Thienthong, Lisa J. Winfield, Jonathan A. Coates, Long Lü,

Bioorganic & Medicinal Chemistry Letters · 2010 · 37 citations · 8 references

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8

Retroviral intasome assembly and inhibition of DNA strand transfer

S. Hare, Saumya Gupta, Eugene Valkov et al. · Nature · 2010 · 666 citations · Full text

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Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection

Vincenzo Summa, Alessia Petrocchi, Fabio Bonelli et al. · Journal of Medicinal Chemistry · 2008 · 634 citations · Full text

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A platform for designing HIV integrase inhibitors. Part 2: A two-metal binding model as a potential mechanism of HIV integrase inhibitors

Takashi Kawasuji, Masahiro Fuji, Tomokazu Yoshinaga et al. · Bioorganic & Medicinal Chemistry · 2006 · 82 citations

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6-Carboxamido-5,4-Hydroxypyrimidinones:  A New Class of Heterocyclic Ligands and Their Evaluation as Gadolinium Chelating Agents

Christopher J. Sunderland, Mauro Botta, Silvio Aime et al. · Inorganic Chemistry · 2001 · 45 citations

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N-Nitroso sultams: on the direction of approach of nucleophiles to the sulfonyl group

Emil H. White, Hyung M. Lim · The Journal of Organic Chemistry · 1987 · 30 citations

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