Concepedia
Statistics
Publications
6
Citations
209
H-Index
Active since
2010
Affiliations
Novita Healthcare (Australia)(Current)
Chinese Academy of Sciences
Shanghai Institute of Organic Chemistry
CSIRO Manufacturing
Division of Materials Science and Engineering
Giang Le is an author at Novita Healthcare (Australia) specializing in drug discovery, ligand binding, and antiretroviral therapy.
Publications per year
2010–2020
Small Molecule Inhibitors of the LEDGF Site of Human Immunodeficiency Virus Integrase Identified by Fragment Screening and Structure Based Design
Thomas S. Peat, David I. Rhodes, Nick Vandegraaff et al. · PLoS ONE · 2012 · 53 citations · Full text
Pharmacy, Medicinal Chemistry, Molecular Biology +17
Structural Basis for a New Mechanism of Inhibition of H I V-1 Integrase Identified by Fragment Screening and Structure-Based Design
David I. Rhodes, Thomas S. Peat, Nick Vandegraaff et al. · Antiviral chemistry & chemotherapy · 2011 · 51 citations
Pharmacy, Biochemistry, Molecular Biology +17
Design of a series of bicyclic HIV-1 integrase inhibitors. Part 1: Selection of the scaffold
E. D. Jones, Nick Vandegraaff, Giang Le et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 37 citations · Full text
Pharmacy, Medicinal Chemistry, Pharmacology +12
Design of a series of bicyclic HIV-1 integrase inhibitors. Part 2: Azoles: Effective metal chelators
Giang Le, Nick Vandegraaff, David I. Rhodes et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 36 citations · Full text
Pharmacy, Chemistry, Medicinal Chemistry +14
Discovery of potent HIV integrase inhibitors active against raltegravir resistant viruses
Giang Le, Nick Vandegraaff, David I. Rhodes et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 20 citations
Life Sciences, Infectious Diseases, Medicinal Chemistry +14
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