Fuk‐Wah Sum

5-Fluoro-2-methyl-<i>N</i>-[4-(5<i>H</i>-pyrrolo[2,1-<i>c</i>]- [1,4]benzodiazepin-10(11<i>H</i>)-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985):  An Orally Active Arginine Vasopressin Antagonist with Selectivity for V₂Receptors

J. Donald Albright, Marvin F. Reich, Efren G. Delos Santos et al. · Journal of Medicinal Chemistry · 1998 · 148 citations · Full text

Altmetric Attention Score, Pharmacotherapy, Experimental Pharmacology +16

Stereoselective synthesis of β-substituted α,β-unsaturated esters by dialkylcuprate coupling to the enol phosphate of β-keto esters

Fuk‐Wah Sum, Larry Weiler · Canadian Journal of Chemistry · 1979 · 105 citations

Corresponding Enol Phosphates, β-Keto Esters, Engineering +13

Indole Cytosolic Phospholipase A₂α Inhibitors: Discovery and in Vitro and in Vivo Characterization of 4-{3-[5-Chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1<i>H</i>-indol-3-yl]propyl}benzoic Acid, Efipladib

John C. McKew, Katherine L. Lee, Marina W. H. Shen et al. · Journal of Medicinal Chemistry · 2008 · 88 citations

Inhibition of Cytosolic Phospholipase A₂α: Hit to Lead Optimization

John C. McKew, Megan A. Foley, Paresh Thakker et al. · Journal of Medicinal Chemistry · 2005 · 76 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Inhibitory Activity +13

Novel (4-Piperidin-1-yl)-phenyl Sulfonamides as Potent and Selective Human β3 Agonists

Baihua Hu, John W. Ellingboe, Stella Han et al. · Bioorganic & Medicinal Chemistry · 2001 · 45 citations

Molecular Pharmacology, Medicinal Chemistry, Pharmaceutical Science +10