Jonathan S. Mason

Discovery of 1,2,4-Triazine Derivatives as Adenosine A_2A Antagonists using Structure Based Drug Design

Miles Congreve, Stephen P. Andrews, A.S. Dore et al. · Journal of Medicinal Chemistry · 2012 · 301 citations · Full text

Combinatorial Chemistry, Compound 4K, Pharmacotherapy +16

Intracellular allosteric antagonism of the CCR9 receptor

Christine Oswald, Mathieu Rappas, James Kean et al. · Nature · 2016 · 270 citations

Inflammation, Signal Transduction, G Protein-coupled Receptor +7

Identification of Novel Adenosine A_2A Receptor Antagonists by Virtual Screening

Christopher J. Langmead, Stephen P. Andrews, Miles Congreve et al. · Journal of Medicinal Chemistry · 2012 · 133 citations · Full text

Enabled Homology Models, Drug Target, Pharmacotherapy +16

Water Network Perturbation in Ligand Binding: Adenosine A_2AAntagonists as a Case Study

Andrea Bortolato, B.G. Tehan, Michael S. Bodnarchuk et al. · Journal of Chemical Information and Modeling · 2013 · 117 citations

Biophysical Mapping of the Adenosine A_2A Receptor

Andrei Zhukov, Stephen P. Andrews, James C. Errey et al. · Journal of Medicinal Chemistry · 2011 · 114 citations · Full text

Molecular Pharmacology, Signal Transduction, Molecular Physiology +15