Andrei Zhukov

Discovery of 1,2,4-Triazine Derivatives as Adenosine A_2A Antagonists using Structure Based Drug Design

Miles Congreve, Stephen P. Andrews, A.S. Dore et al. · Journal of Medicinal Chemistry · 2012 · 301 citations · Full text

Combinatorial Chemistry, Compound 4K, Pharmacotherapy +16

Structural insight into allosteric modulation of protease-activated receptor 2

R.K. Cheng, Cédric Fiez-Vandal, Oliver Schlenker et al. · Nature · 2017 · 246 citations

Signal Transduction, Biochemistry, G Protein-coupled Receptor +6

The properties of thermostabilised G protein-coupled receptors (StaRs) and their use in drug discovery

N.J. Robertson, Ali Jazayeri, James C. Errey et al. · Neuropharmacology · 2010 · 158 citations

Drug Target, Biochemistry, G Protein-coupled Receptor +5

Identification of Novel Adenosine A_2A Receptor Antagonists by Virtual Screening

Christopher J. Langmead, Stephen P. Andrews, Miles Congreve et al. · Journal of Medicinal Chemistry · 2012 · 133 citations · Full text

Enabled Homology Models, Drug Target, Pharmacotherapy +16

Biophysical Mapping of the Adenosine A_2A Receptor

Andrei Zhukov, Stephen P. Andrews, James C. Errey et al. · Journal of Medicinal Chemistry · 2011 · 114 citations · Full text

Molecular Pharmacology, Signal Transduction, Molecular Physiology +15