Françoise Gellibert

Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains

Chun‐wa Chung, Hervé Coste, Julia H. White et al. · Journal of Medicinal Chemistry · 2011 · 335 citations · Full text

Life Sciences, Medicinal Chemistry, Molecular Biology +17

Identification of 1,5-Naphthyridine Derivatives as a Novel Series of Potent and Selective TGF-β Type I Receptor Inhibitors

Françoise Gellibert, James M. Woolven, Marie-Hélène Fouchet et al. · Journal of Medicinal Chemistry · 2004 · 222 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Oral administration of GW788388, an inhibitor of TGF-β type I and II receptor kinases, decreases renal fibrosis

Maj Petersen, Midory Thorikay, Martijn Deckers et al. · Kidney International · 2007 · 214 citations · Full text

Medicine, Pharmacology, Pharmacotherapy +13

Identification of a novel series of BET family bromodomain inhibitors: Binding mode and profile of I-BET151 (GSK1210151A)

Jonathan T. Seal, Yann Lamotte, Frédéric Donche et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 213 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +16

Inhibition of TGF‐<i>β</i> signaling by an ALK5 inhibitor protects rats from dimethylnitrosamine‐induced liver fibrosis

Anne‐Charlotte de Gouville, Valérie Boullay, Gaël Krysa et al. · British Journal of Pharmacology · 2005 · 165 citations · Full text

Life Sciences, Molecular Biology, Pharmacology +14