Steven Ronkin

Novel Dual-Targeting Benzimidazole Urea Inhibitors of DNA Gyrase and Topoisomerase IV Possessing Potent Antibacterial Activity: Intelligent Design and Evolution through the Judicious Use of Structure-Guided Design and Stucture−Activity Relationships

Paul S. Charifson, Anne‐Laure Grillot, Trudy H. Grossman et al. · Journal of Medicinal Chemistry · 2008 · 222 citations · Full text

Bioorganic Chemistry, Antibacterial Activity, Molecular Biology +23

Discovery of pyrazolthiazoles as novel and potent inhibitors of bacterial gyrase

Steven Ronkin, Michael C. Badia, S.F. Bellon et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 104 citations

Antifungal Agent, Medicine, Bacterial Gyrase +9

Discovery of Potent, Selective Triazolothiadiazole-Containing c-Met Inhibitors

Qing Tang, Alex M. Aronov, David D. Deininger et al. · ACS Medicinal Chemistry Letters · 2021 · 13 citations · Full text

Discovery of Novel, Orally Bioavailable Pyrimidine Ether-Based Inhibitors of ELOVL1

Michael J. Boyd, Philip N. Collier, Michael P. Clark et al. · Journal of Medicinal Chemistry · 2021 · 13 citations · Full text

Discovery of Novel Thiophene-Based, Thumb Pocket 2 Allosteric Inhibitors of the Hepatitis C NS5B Polymerase with Improved Potency and Physicochemical Profiles

John J. Court, Carl Poisson, Andrzej Ardzinski et al. · Journal of Medicinal Chemistry · 2016 · 12 citations · Full text

Immunology, Allosteric Inhibitors, Antiviral Drug +19