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Kristin M. Riching, Sarah D. Mahan, Cesear Corona, +5

ACS Chemical Biology

Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement

James D. Vasta, Cesear Corona, Jennifer Wilkinson, +25

Cell chemical biology

Drug TargetWide-spectrum Kinase ProfilingKinase InhibitorsCytoskeletonCellular Physiology +18

Synthetic Estrogen Derivatives Demonstrate the Functionality of Intracellular GPR30

Chetana M. Revankar, Hugh Mitchell, Angela S. Field, +6

ACS Chemical Biology

Selective JAK3 Inhibitors with a Covalent Reversible Binding Mode Targeting a New Induced Fit Binding Pocket

Michael Förster, A. Chaikuad, Silke M. Bauer, +8

Cell chemical biology

Discovery of a selective inhibitor of doublecortin like kinase 1

Fleur M. Ferguson, Behnam Nabet, Srivatsan Raghavan, +34

Nature Chemical Biology

MedicineReceptor Tyrosine KinaseKinase 1PharmacologyCell Biology +3

Quantifying CDK inhibitor selectivity in live cells

Carrow I. Wells, James D. Vasta, Cesear Corona, +14

Nature Communications

KRAS is vulnerable to reversible switch-II pocket engagement in cells

James D. Vasta, D. Matthew Peacock, Qinheng Zheng, +9

Nature Chemical Biology

Bisphenol A Directly Targets Tubulin to Disrupt Spindle Organization in Embryonic and Somatic Cells

Olivia George, Bj K. Bryant, Chinnasamy Ramesh, +3

ACS Chemical Biology

GeneticsCell CultureCytoskeletonReproductive BiologyCellular Physiology +17

NanoClick: A High Throughput, Target-Agnostic Peptide Cell Permeability Assay

Andrea Peier, Lan Ge, N. Boyer, +22

ACS Chemical Biology

Homogeneous plate based antibody internalization assay using pH sensor fluorescent dye

Nidhi Nath, Becky Godat, Chad Zimprich, +4

Journal of Immunological Methods

Immunocytochemical TechniqueEngineeringBiosensing SystemsHomogeneous PlateMedicine +13