Anna Waszkiewicz

An Orally Active TRPV4 Channel Blocker Prevents and Resolves Pulmonary Edema Induced by Heart Failure

Kevin S. Thorneloe, Mui Cheung, Weike Bao et al. · Science Translational Medicine · 2012 · 336 citations

Medicine, Cardiology, Pharmacotherapy +10

The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore

David G. Washburn, Dennis A. Holt, Jason W. Dodson et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 58 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

A High-Throughput Dose-Response Cellular Thermal Shift Assay for Rapid Screening of Drug Target Engagement in Living Cells, Exemplified Using SMYD3 and IDO1

Dean E. McNulty, William G. Bonnette, Hongwei Qi et al. · SLAS DISCOVERY · 2017 · 51 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Dexamethasone-dependent modulation of cyclic GMP synthesis in podocytes

Barbara Lewko, Anna Waszkiewicz, Anna Maryn et al. · Molecular and Cellular Biochemistry · 2015 · 15 citations · Full text

Medicine, Nephrology, Physiology +13

High-Throughput Screening and Triage Assays Identify Small Molecules Targeting c-MYC in Cancer Cells

Lorena A. Kallal, Anna Waszkiewicz, Jon‐Paul Jaworski et al. · SLAS DISCOVERY · 2021 · 10 citations · Full text

Medicine, Molecular Biology, Oncology +17