Dariusz Wódka

Identification of 2-(4-Benzyloxyphenyl)-<i>N</i>- [1-(2-pyrrolidin-1-yl-ethyl)-1<i>H</i>-indazol-6-yl]acetamide, an Orally Efficacious Melanin-Concentrating Hormone Receptor 1 Antagonist for the Treatment of Obesity

Andrew J. Souers, Ju Gao, Michael E. Brune et al. · Journal of Medicinal Chemistry · 2005 · 88 citations · Full text

Discovery and Metabolic Stabilization of Potent and Selective 2-Amino-<i>N</i>-(adamant-2-yl) Acetamide 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors

Jeffrey J. Rohde, Marina Pliushchev, Bryan K. Sorensen et al. · Journal of Medicinal Chemistry · 2006 · 76 citations · Full text

Medicinal Chemistry, Pharmacological Study, Biochemistry +11

Optimization of Chromone-2-carboxamide Melanin Concentrating Hormone Receptor 1 Antagonists:  Assessment of Potency, Efficacy, and Cardiovascular Safety

J.A. Lynch, Jennifer C. Freeman, Andrew S. Judd et al. · Journal of Medicinal Chemistry · 2006 · 48 citations · Full text

Metabolic Syndrome, Medicinal Chemistry, Distinct Series +14

Discovery and Characterization of Aminopiperidinecoumarin Melanin Concentrating Hormone Receptor 1 Antagonists

Philip R. Kym, Rajesh Iyengar, Andrew J. Souers et al. · Journal of Medicinal Chemistry · 2005 · 48 citations · Full text

Cardiovascular Pharmacology, Pharmacotherapy, Metabolic Syndrome +17

Synthesis and evaluation of urea-based indazoles as melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity

Andrew J. Souers, Ju Gao, Dariusz Wódka et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 44 citations · Full text

Urea-based Indazoles, Medicine, Physiology +4