Concepedia

Development of triazolothiadiazine derivatives as highly potent tubulin polymerization inhibitors: Structure-activity relationship, in vitro and in vivo study

Weifeng Ma, Peng Chen, Xian‐Sen Huo, Yufeng Ma, Yanhong Li, Peng-Cheng Diao, Fang Yang, Shengquan Zheng, Meng‐Jin Hu, Wen‐Wei You,

European Journal of Medicinal Chemistry · 2020 · 46 citations · 37 references

DOI

Concepts

References

37

Insight into tubulin regulation from a complex with colchicine and a stathmin-like domain

Raimond B. G. Ravelli, Benoı̂t Gigant, Patrick A. Curmi et al. · Nature · 2004 · 1.6K citations

, , +14

Combretastatin A-4, an agent that displays potent and selective toxicity toward tumor vasculature.

G. Dark, S A Hill, Vivien E. Prise et al. · PubMed · 1997 · 624 citations

, , +13

Anti-vascular approaches to solid tumour therapy: evaluation of combretastatin A4 phosphate.

David J. Chaplin, George R. Pettit, S A Hill · PubMed · 1999 · 252 citations

, , +17

Class III β-tubulin expression and in vitro resistance to microtubule targeting agents

Chloé Stengel, Stephen T. Newman, Mathew P. Leese et al. · British Journal of Cancer · 2009 · 191 citations · Full text

, , +16

Differential cytotoxicity of Combretastatins A1 and A4 in two daunorubicin-resistant P388 cell lines

Alan T. McGown, Brian W. Fox · Cancer Chemotherapy and Pharmacology · 1990 · 138 citations

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