An improved procedure for the regiospecific synthesis of electron deficient 4- and 6-substituted isatins

Design, Synthesis, and Evaluation of Nonpeptidic Inhibitors of Human Rhinovirus 3C Protease

Stephen E. Webber, Jayashree Tikhe, Stephen T. Worland et al. · Journal of Medicinal Chemistry · 1996 · 145 citations · Full text

Life Sciences, Biochemistry, Medicinal Chemistry +16

A general method for the synthesis of isatins

Paul G. Gassman, Berkeley W. Cue, Tien‐Yau Luh · The Journal of Organic Chemistry · 1977 · 91 citations

Natural Sciences, Chemistry, Analytical Chemistry +5

Antiinflammatory agents. 3. Synthesis and pharmacological evaluation of 2-amino-3-benzoylphenylacetic acid and analogs

David A. Walsh, H. W. MORAN, Dwight A. Shamblee et al. · Journal of Medicinal Chemistry · 1984 · 75 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +8

A general method for the synthesis of isatins: Preparation of regiospecifically functionalized isatins from anilines

Piyasena Hewawasam, Nicholas A. Meanwell · Tetrahedron Letters · 1994 · 69 citations

Pharmacy, Medicinal Chemistry, Synthetic Medicinal Chemistry +2

4-Substituted-3-phenylquinolin-2(1<i>H</i>)-ones:  Acidic and Nonacidic Glycine Site<i>N</i>-Methyl-<scp>d</scp>-aspartate Antagonists with<i>in</i><i>Vivo</i>Activity

Robert W. Carling, Paul D. Leeson, Kevin W. Moore et al. · Journal of Medicinal Chemistry · 1997 · 67 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14